Uso: Declínio da função sexual; Transtorno sexual não orgânico, Pacientes de pronto-socorro.
É o primeiro composto desenvolvido especialmente para o tratamento da ejaculação precoce (Educação Física) em homens 18-64 anos. funciona inibindo o transportador de serotonina, aumentando a ação da serotonina na fenda pós-sináptica, e como consequência promovendo atraso ejaculatório. Como membro do inibidor seletivo da recaptação da serotonina (ISRS) família, was initially created as an antidepressant. No entanto, unlike other SSRIs, is absorbed and eliminated rapidly in the body. Its fast acting property makes it suitable for the treatment of PE but not as an antidepressant.
It is as a new fast SSRI, a short half life, a selective 5 – HT reuptake inhibitor (ISRS), for the treatment of premature ejaculation and erectile dysfunction. is a selective 5 – HT reuptake inhibitor (ISRS), such drugs widely used to treat depression and related affective disorders.
This ingredients belongs to phosphodiesterase type 5 of this kind of inhibitor. When sexuelle erregung, neurone of NANC and nitrogen oxide in endothelial cells synthase and catalyse L-arginine to synthetize nitrogen oxide, which activate guanosine to synthesis increase, then lead cavernous body of penis smooth muscle and artery of penis into relaxation, blood into penis sponge sinus, make penis erect.